{"id":1094,"date":"2020-07-09T21:39:11","date_gmt":"2020-07-09T19:39:11","guid":{"rendered":"https:\/\/covid.si\/?p=1094"},"modified":"2020-11-02T21:19:27","modified_gmt":"2020-11-02T20:19:27","slug":"misija-4-iskanje-inhibitorjev-encima-dhodh","status":"publish","type":"post","link":"https:\/\/covid.si\/en\/misija-4-iskanje-inhibitorjev-encima-dhodh\/","title":{"rendered":"MI 4:  Zavrimo COVID-19 &#8211; Zaviralci DHODH"},"content":{"rendered":"\t\t<div data-elementor-type=\"wp-post\" data-elementor-id=\"1094\" class=\"elementor elementor-1094\" data-elementor-post-type=\"post\">\n\t\t\t\t\t\t<section data-particle_enable=\"false\" data-particle-mobile-disabled=\"false\" class=\"elementor-section elementor-top-section elementor-element elementor-element-3b8a885 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"3b8a885\" data-element_type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-100 elementor-top-column elementor-element elementor-element-3be75e6\" data-id=\"3be75e6\" data-element_type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-4a0ec66 elementor-widget elementor-widget-theme-post-title elementor-page-title elementor-widget-heading\" data-id=\"4a0ec66\" data-element_type=\"widget\" data-widget_type=\"theme-post-title.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t<h2 class=\"elementor-heading-title elementor-size-default\">MI 4:  Zavrimo COVID-19 &#8211; Zaviralci DHODH<\/h2>\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<div class=\"elementor-element elementor-element-e8d41fc elementor-widget-divider--view-line elementor-widget elementor-widget-divider\" data-id=\"e8d41fc\" data-element_type=\"widget\" data-widget_type=\"divider.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<div class=\"elementor-divider\">\n\t\t\t<span class=\"elementor-divider-separator\">\n\t\t\t\t\t\t<\/span>\n\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section data-particle_enable=\"false\" data-particle-mobile-disabled=\"false\" class=\"elementor-section elementor-top-section elementor-element elementor-element-b2d1c2b elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"b2d1c2b\" data-element_type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-bc5d83e\" data-id=\"bc5d83e\" data-element_type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-e3c3d1d elementor-widget elementor-widget-text-editor\" data-id=\"e3c3d1d\" data-element_type=\"widget\" data-widget_type=\"text-editor.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t<h5>STATUS MISIJE:\u00a0<strong>REZULTATI V OBDELAVI<\/strong><\/h5><div><strong>\u00a0<\/strong><\/div><h5>NA\u010cRT MISIJE:<strong> Domen Oblak\u00a0in dr. \u010crtomir Podlipnik<\/strong><\/h5><h5>\u0160tevilo tar\u010d: 6<\/h5><h5>Oznake tar\u010d: 35<strong>-40<\/strong><\/h5><h5>\u0160tevilo spojin: preko\u00a0<strong>10 M<\/strong><\/h5><h5>Skupaj sidrano 6<b>0 M<\/b>\u00a0spojin<\/h5><h5>Trajanje misije: 27<strong>.05.2020 &#8211;<\/strong><\/h5><h5>Rezultati: <strong>v obdelavi<\/strong><\/h5>\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-999c372\" data-id=\"999c372\" data-element_type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-de98b41 elementor-widget elementor-widget-image\" data-id=\"de98b41\" data-element_type=\"widget\" data-widget_type=\"image.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t\t\t\t\t\t\t<img fetchpriority=\"high\" decoding=\"async\" width=\"848\" height=\"228\" src=\"https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/dhodh.png\" class=\"attachment-large size-large wp-image-1097\" alt=\"\" srcset=\"https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/dhodh.png 848w, https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/dhodh-300x81.png 300w, https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/dhodh-768x206.png 768w, https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/dhodh-720x194.png 720w, https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/dhodh-350x94.png 350w\" sizes=\"(max-width: 848px) 100vw, 848px\" \/>\t\t\t\t\t\t\t\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section data-particle_enable=\"false\" data-particle-mobile-disabled=\"false\" class=\"elementor-section elementor-top-section elementor-element elementor-element-8837460 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"8837460\" data-element_type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-100 elementor-top-column elementor-element elementor-element-0df1c58\" data-id=\"0df1c58\" data-element_type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-a3cd1b4 elementor-widget elementor-widget-text-editor\" data-id=\"a3cd1b4\" data-element_type=\"widget\" data-widget_type=\"text-editor.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t<p><strong>Seznam tar\u010d:<\/strong><\/p><p><strong>#35 <\/strong><a href=\"https:\/\/www.rcsb.org\/structure\/4iGH\"><strong>4igh<\/strong><\/a><strong> \u2013 <\/strong>High resolution crystal structure of human dihydroorotate dehydrogenase bound with 4-quinoline carboxylic acid analog<\/p><p><strong>#36 <\/strong><a href=\"https:\/\/www.rcsb.org\/structure\/4JTU\"><strong>4jtu<\/strong><\/a><strong> &#8211; <\/strong>Crystal structure of human dihydroorotate dehydrogenase (DHODH) with brequinar analogue<\/p><p><strong>#37 <\/strong><a href=\"https:\/\/www.rcsb.org\/structure\/4oqv\"><strong>4oqv<\/strong><\/a><strong> &#8211; <\/strong>High resolution crystal structure of human dihydroorotate dehydrogenase bound with DSM338 (N-[3,5-difluoro-4-(trifluoromethyl)phenyl]-5-methyl-2-(trifluoromethyl)[1,2,4]triazolo[1,5-a]pyrimidin-7-amine)<\/p><p><strong>#38 <\/strong><a href=\"https:\/\/www.rcsb.org\/structure\/3I65\"><strong>3i65<\/strong><\/a><strong> &#8211; <\/strong>Plasmodium falciparum dihydroorotate dehydrogenase bound with triazolopyrimidine-based inhibitor DSM1<\/p><p><strong>#39 <\/strong><a href=\"https:\/\/www.rcsb.org\/structure\/4cq8\"><strong>4cq8<\/strong><\/a><strong> &#8211; <\/strong>Plasmodium falciparum dihydroorotate dehydrogenase (DHODH) in complex with Genz-669178<\/p><p><strong>#40 <\/strong><a href=\"https:\/\/www.rcsb.org\/structure\/4rx0\"><strong>4rx0<\/strong><\/a><strong> &#8211; <\/strong>Crystal structure of Plasmodium falciparum dihydroorotate dehydrogenase bound with Inhibitor DSM265<\/p><p><u>OPIS MISIJE:<\/u>\u00a0<\/p><p>REFERENCE:<\/p><p><span style=\"color: #494949; font-family: 'Open Sans', 'Myriad Pro', 'Helvetica Neue', Helvetica, Arial, sans-serif; font-size: 14px;\">Xiong R, Zhang L, Li S, et al. Novel and potent inhibitors targeting DHODH, a rate-limiting enzyme in de novo pyrimidine biosynthesis, are broad-spectrum antiviral against RNA viruses including newly emerged coronavirus SARS-CoV-2. bioRxiv; 2020. DOI: 10.1101\/2020.03.11.983056.<\/span><\/p><p><span style=\"color: #494949; font-family: 'Open Sans', 'Myriad Pro', 'Helvetica Neue', Helvetica, Arial, sans-serif; font-size: 14px;\">\u00a0<\/span><\/p><p>\u00a0<\/p>\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<\/div>\n\t\t","protected":false},"excerpt":{"rendered":"<p>STATUS MISIJE:&nbsp;REZULTATI V OBDELAVI &nbsp; NA\u010cRT MISIJE: Domen Oblak&nbsp;in dr. \u010crtomir Podlipnik \u0160tevilo tar\u010d: 6 Oznake tar\u010d: 35-40 \u0160tevilo spojin: [&hellip;]<\/p>\n","protected":false},"author":2,"featured_media":0,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[10],"tags":[58,4,56,61,59,57,55,60],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v22.5 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>MI 4: Zavrimo COVID-19 - Zaviralci DHODH - COVID.SI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/covid.si\/misija-4-iskanje-inhibitorjev-encima-dhodh\/\" \/>\n<meta property=\"og:locale\" content=\"en_GB\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"MI 4: Zavrimo COVID-19 - Zaviralci DHODH - COVID.SI\" \/>\n<meta property=\"og:description\" content=\"STATUS MISIJE:&nbsp;REZULTATI V OBDELAVI &nbsp; 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