{"id":1105,"date":"2020-07-10T10:56:40","date_gmt":"2020-07-10T08:56:40","guid":{"rendered":"https:\/\/covid.si\/?p=1105"},"modified":"2020-11-02T21:14:48","modified_gmt":"2020-11-02T20:14:48","slug":"misija-5-inhibitorji-virusne-proteaze-plpro-sars-cov-sars-cov2","status":"publish","type":"post","link":"https:\/\/covid.si\/en\/misija-5-inhibitorji-virusne-proteaze-plpro-sars-cov-sars-cov2\/","title":{"rendered":"MI5: Zavrimo COVID-19 z inhibicijo virusne PL proteaze"},"content":{"rendered":"\t\t<div data-elementor-type=\"wp-post\" data-elementor-id=\"1105\" class=\"elementor elementor-1105\" data-elementor-post-type=\"post\">\n\t\t\t\t\t\t<section data-particle_enable=\"false\" data-particle-mobile-disabled=\"false\" class=\"elementor-section elementor-top-section elementor-element elementor-element-3b8a885 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"3b8a885\" data-element_type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-100 elementor-top-column elementor-element elementor-element-3be75e6\" data-id=\"3be75e6\" data-element_type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-4a0ec66 elementor-widget elementor-widget-theme-post-title elementor-page-title elementor-widget-heading\" data-id=\"4a0ec66\" data-element_type=\"widget\" data-widget_type=\"theme-post-title.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t<h2 class=\"elementor-heading-title elementor-size-default\">MI5: Zavrimo COVID-19 z inhibicijo virusne PL proteaze<\/h2>\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<div class=\"elementor-element elementor-element-e8d41fc elementor-widget-divider--view-line elementor-widget elementor-widget-divider\" data-id=\"e8d41fc\" data-element_type=\"widget\" data-widget_type=\"divider.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t<div class=\"elementor-divider\">\n\t\t\t<span class=\"elementor-divider-separator\">\n\t\t\t\t\t\t<\/span>\n\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section data-particle_enable=\"false\" data-particle-mobile-disabled=\"false\" class=\"elementor-section elementor-top-section elementor-element elementor-element-b2d1c2b elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"b2d1c2b\" data-element_type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-bc5d83e\" data-id=\"bc5d83e\" data-element_type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-e3c3d1d elementor-widget elementor-widget-text-editor\" data-id=\"e3c3d1d\" data-element_type=\"widget\" data-widget_type=\"text-editor.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t<h5>STATUS MISIJE:\u00a0<strong>REZULTATI V OBDELAVI<\/strong><\/h5><div><strong>\u00a0<\/strong><\/div><h5>NA\u010cRT MISIJE:<strong>\u00a0 dr. \u010crtomir Podlipnik in Ga\u0161per Tom\u0161i\u010d<\/strong><\/h5><h5>\u0160tevilo tar\u010d: 8<\/h5><h5>Oznake tar\u010d: 41<strong>-48<\/strong><\/h5><h5>\u0160tevilo spojin: preko\u00a0<strong>10 M<\/strong><\/h5><h5>Skupaj sidrano 8<b>0 M<\/b>\u00a0spojin<\/h5><h5>Trajanje misije: 16<strong>.06.2020 &#8211;<\/strong><\/h5><h5>Rezultati: <strong>v obdelavi<\/strong><\/h5>\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t<div class=\"elementor-column elementor-col-50 elementor-top-column elementor-element elementor-element-999c372\" data-id=\"999c372\" data-element_type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-de98b41 elementor-widget elementor-widget-image\" data-id=\"de98b41\" data-element_type=\"widget\" data-widget_type=\"image.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t\t\t\t\t\t\t<img fetchpriority=\"high\" decoding=\"async\" width=\"1024\" height=\"452\" src=\"https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/PLPro46.png\" class=\"attachment-large size-large wp-image-1107\" alt=\"\" srcset=\"https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/PLPro46.png 1024w, https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/PLPro46-300x132.png 300w, https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/PLPro46-768x339.png 768w, https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/PLPro46-720x318.png 720w, https:\/\/covid.si\/wp-content\/uploads\/2020\/07\/PLPro46-350x154.png 350w\" sizes=\"(max-width: 1024px) 100vw, 1024px\" \/>\t\t\t\t\t\t\t\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<section data-particle_enable=\"false\" data-particle-mobile-disabled=\"false\" class=\"elementor-section elementor-top-section elementor-element elementor-element-8837460 elementor-section-boxed elementor-section-height-default elementor-section-height-default\" data-id=\"8837460\" data-element_type=\"section\">\n\t\t\t\t\t\t<div class=\"elementor-container elementor-column-gap-default\">\n\t\t\t\t\t<div class=\"elementor-column elementor-col-100 elementor-top-column elementor-element elementor-element-0df1c58\" data-id=\"0df1c58\" data-element_type=\"column\">\n\t\t\t<div class=\"elementor-widget-wrap elementor-element-populated\">\n\t\t\t\t\t\t<div class=\"elementor-element elementor-element-a3cd1b4 elementor-widget elementor-widget-text-editor\" data-id=\"a3cd1b4\" data-element_type=\"widget\" data-widget_type=\"text-editor.default\">\n\t\t\t\t<div class=\"elementor-widget-container\">\n\t\t\t\t\t\t\t<p><strong>Seznam tar\u010d:<\/strong><\/p><p><strong>#41 <a href=\"https:\/\/www.rcsb.org\/structure\/2fe8\">2fe8<\/a> \u2013 <\/strong>SARS coronavirus papain-like protease: structure of a viral deubiquitinating enzyme<\/p><p><strong>#42 <a href=\"https:\/\/www.rcsb.org\/structure\/3mp2\">3mp2<\/a> &#8211; C<\/strong>rystal structure of transmissible gastroenteritis virus papain-like protease 1<\/p><p><strong>#43 <a href=\"https:\/\/www.rcsb.org\/structure\/4ow0\">4ow0<\/a>&#8211; <\/strong>X-Ray Structural and Biological Evaluation of a Series of Potent and Highly Selective Inhibitors of Human Coronavirus Papain-Like Proteases<\/p><p><strong>#44 <a href=\"https:\/\/www.rcsb.org\/structure\/6w9c\">6w9c<\/a>&#8211; <\/strong>The crystal structure of papain-like protease of SARS CoV-2<\/p><p><strong>#45 <a href=\"https:\/\/www.rcsb.org\/structure\/6wrh\">6wrh<\/a> &#8211;<\/strong> The crystal structure of Papain-Like Protease of SARS CoV-2 , C111S mutant<\/p><p><strong>#46 <a href=\"https:\/\/www.rcsb.org\/structure\/6wuu\">6wuu<\/a> &#8211; <\/strong>Crystal structure of the SARS CoV-2 Papain-like protease in complex with peptide inhibitor VIR250<\/p><p><strong>#47 <a href=\"https:\/\/www.rcsb.org\/structure\/6wx4\">6wx4<\/a> &#8211; <\/strong>Crystal structure of the SARS CoV-2 Papain-like protease in complex with peptide inhibitor VIR251<\/p><p><strong>#48 <a href=\"https:\/\/www.rcsb.org\/structure\/6wzu\">6wzu<\/a> &#8211; <\/strong>The crystal structure of Papain-Like Protease of SARS CoV-2 , P3221 space group<\/p><p>\u00a0<\/p><p><u>OPIS MISIJE:<\/u>\u00a0<\/p><p>REFERENCE:<\/p><p><a href=\"https:\/\/doi.org\/10.1016\/j.antiviral.2014.12.015\">https:\/\/doi.org\/10.1016\/j.antiviral.2014.12.015<\/a><\/p><p><a href=\"https:\/\/www.drugtargetreview.com\/news\/63123\/naphthalene-based-plpro-inhibitors-show-potential-as-covid-19-therapeutics\/\">https:\/\/www.drugtargetreview.com\/news\/63123\/naphthalene-based-plpro-inhibitors-show-potential-as-covid-19-therapeutics\/<\/a><\/p><p><a id=\"dest_link\" style=\"border-bottom-color: #112e51; border-bottom-style: solid; border-bottom-width: 1px; box-sizing: border-box; color: #1a3d85; cursor: pointer; font-family: &amp;quot; source sans pro&amp;quot;,&amp;quot;helvetica neue&amp;quot;,&amp;quot;helvetica&amp;quot;,&amp;quot;roboto&amp;quot;,&amp;quot;arial&amp;quot;,sans-serif; font-size: 15px; font-style: normal; font-variant: normal; font-weight: 400; letter-spacing: normal; orphans: 2; text-align: left; text-decoration: none; text-indent: 0px; text-transform: none; transition-delay: 0s; transition-duration: 0.1s; transition-property: color; transition-timing-function: linear; -webkit-text-stroke-width: 0px; white-space: normal; word-spacing: 0px;\" href=\"https:\/\/doi.org\/10.1101\/2020.02.23.20026690\">https:\/\/doi.org\/10.1101\/2020.02.23.20026690<\/a><b><\/b><i><\/i><u><\/u><\/p><p>\u00a0<\/p><p><span style=\"color: #494949; font-family: 'Open Sans', 'Myriad Pro', 'Helvetica Neue', Helvetica, Arial, sans-serif; font-size: 14px;\">\u00a0<\/span><\/p><p>\u00a0<\/p>\t\t\t\t\t\t<\/div>\n\t\t\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/div>\n\t\t\t\t\t<\/div>\n\t\t<\/section>\n\t\t\t\t<\/div>\n\t\t","protected":false},"excerpt":{"rendered":"<p>STATUS MISIJE:&nbsp;REZULTATI V OBDELAVI &nbsp; NA\u010cRT MISIJE:&nbsp; dr. \u010crtomir Podlipnik in Ga\u0161per Tom\u0161i\u010d \u0160tevilo tar\u010d: 8 Oznake tar\u010d: 41-48 \u0160tevilo [&hellip;]<\/p>\n","protected":false},"author":2,"featured_media":0,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[10],"tags":[52,51,44,48,42,49,43,50,54,53],"yoast_head":"<!-- This site is optimized with the 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